smiles
stringlengths
6
253
ki
float64
0
2,570,395,783B
receptor
stringlengths
2
90
source
stringclasses
243 values
CN1CCC(=C2C3=CC=CC=C3C=CC4=CC=CC=C42)CC1
99
5-HT1A
CORTEX
CN1CCC(=C2C3=CC=CC=C3C=CC4=CC=CC=C42)CC1
110
5-HT1A
CORTEX
CN1CCC(=C2C3=CC=CC=C3C=CC4=CC=CC=C42)CC1
112.9
5-HT1A
CORTEX
CN1CCC(=C2C3=CC=CC=C3C=CC4=CC=CC=C42)CC1
355
5-HT1A
CORTEX
CN1CCC(=C2C3=CC=CC=C3C=CC4=CC=CC=C42)CC1
355
5-HT1A
CORTEX
CN1CCC(=C2C3=CC=CC=C3C=CC4=CC=CC=C42)CC1
759.89
5-HT1A
HIPPOCAMPUS
CC1=C(C(=CC=C1)N2CCNCC2)C
622.48
5-HT1A
HIPPOCAMPUS
null
10,000
5-HT1A
HIPPOCAMPUS
COC1=CC=CC=C1N2CCNCC2
130.37
5-HT1A
HIPPOCAMPUS
null
206.13
5-HT1A
HIPPOCAMPUS
null
366.52
5-HT1A
HIPPOCAMPUS
null
0.29
5-HT1A
CORTEX
null
0.29
5-HT1A
CORTEX
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
14
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
14
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
15
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
15
5-HT1A
CORTEX
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
15.8
5-HT1A
CORTEX
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
17.78
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
20
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
20.89
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
22.94
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
23.4
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
26.3
5-HT1A
CORTEX
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
26.3
5-HT1A
CORTEX
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
31.19
5-HT1A
HIPPOCAMPUS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
74.1
5-HT1A
CELLS
C1CCC2(C1)CC(=O)N(C(=O)C2)CCCCN3CCN(CC3)C4=NC=CC=N4
97
5-HT1A
CELLS
CC(C)(C)C1(CCN2CC3C4=CC=CC=C4CCC5=C3C(=CC=C5)C2C1)O
6.6
5-HT1A
CELLS
CC(C)(C)C1(CCN2CC3C4=CC=CC=C4CCC5=C3C(=CC=C5)C2C1)O
9.5
5-HT1A
CELLS
CC(C)(C)NCC(COC1=CC=CC2=C1C=C(N2)C#N)O
5.37
5-HT1A
CORTEX
CC(C)(C)NCC(COC1=CC=CC2=C1C=C(N2)C#N)O
53.7
5-HT1A
CORTEX
CNCCCN1C2=CC=CC=C2CCC3=CC=CC=C31
10,000
5-HT1A
HIPPOCAMPUS
CN1C(=O)CN=C(C2=C1C=CC(=C2)Cl)C3=CC=CC=C3
10,000
5-HT1A
HIPPOCAMPUS
CC(C)CC1C(=O)N2CCCC2C3(N1C(=O)C(O3)(C(C)C)NC(=O)C4CC5C(CC6=CNC7=CC=CC5=C67)N(C4)C)O
0.09
5-HT1A
CORTEX
CC1(C(=O)N2C(C(=O)N3CCCC3C2(O1)O)CC4=CC=CC=C4)NC(=O)C5CC6C(CC7=CNC8=CC=CC6=C78)N(C5)C
1.23
5-HT1A
CORTEX
CC1(C(=O)N2C(C(=O)N3CCCC3C2(O1)O)CC4=CC=CC=C4)NC(=O)C5CC6C(CC7=CNC8=CC=CC6=C78)N(C5)C
19
5-HT1A
CORTEX
CC(=O)OC1C(SC2=CC=CC=C2N(C1=O)CCN(C)C)C3=CC=C(C=C3)OC.Cl
10,000
5-HT1A
CORTEX
CN(C)CCC1=CNC2=CC=CC=C21
119.51
5-HT1A
CORTEX
CN(C)CCC1=CNC2=CC=CC=C21
140.74
5-HT1A
HIPPOCAMPUS
CN(C)CCC1=CNC2=CC=CC=C21
245
5-HT1A
CORTEX
CC(CC1=CC(=C(C=C1OC)Br)OC)N
3,770
5-HT1A
HIPPOCAMPUS
CC(CC1=CC(=C(C=C1OC)Br)OC)N
6,326.73
5-HT1A
CORTEX
CC(CC1=CC(=C(C=C1OC)Br)OC)N
3,770
5-HT1A
HIPPOCAMPUS
CC(C1=CC=CC2=NC3=C(C=CC=C3N=C21)C(=O)O)OC(=O)C(CO)OC
2,332
5-HT1A
HIPPOCAMPUS
null
4,041
5-HT1A
HIPPOCAMPUS
null
4,178
5-HT1A
HIPPOCAMPUS
CCC1=CC(=C(C=C1OC)CC(C)N)OC.Cl
3,930
5-HT1A
HIPPOCAMPUS
CC(CC1=CC(=C(C=C1OC)I)OC)N
2,355
5-HT1A
HIPPOCAMPUS
CC1(CC(=O)N(C(=O)C1)CCCCN2CCN(CC2)C3=NC=CC=N3)C.Cl
70
5-HT1A
HIPPOCAMPUS
CC1(CC(=O)N(C(=O)C1)CCCCN2CCN(CC2)C3=NC=CC=N3)C.Cl
89.1
5-HT1A
CORTEX
C1CN(CCC1(C2=CC=C(C=C2)Cl)O)CCCC(=O)C3=CC=C(C=C3)F
346.2
5-HT1A
CORTEX
C1CN(CCC1(C2=CC=C(C=C2)Cl)O)CCCC(=O)C3=CC=C(C=C3)F
2,761.11
5-HT1A
HIPPOCAMPUS
C1CN(CCC1(C2=CC=C(C=C2)Cl)O)CCCC(=O)C3=CC=C(C=C3)F
2,800
5-HT1A
CORTEX
C1CN(CCC1(C2=CC=C(C=C2)Cl)O)CCCC(=O)C3=CC=C(C=C3)F
4,790
5-HT1A
CORTEX
C1=C(NC=N1)CCN
6,011
5-HT1A
CELLS
C1=C(NC=N1)CCN
10,000
5-HT1A
HIPPOCAMPUS
C1=C(NC=N1)CCN
10,000
5-HT1A
CORTEX
CN1C2CCC1CC(C2)OC(=O)C3=CNC4=CC=CC=C43
1,788
5-HT1A
CELLS
CN1C2CCC1CC(C2)OC(=O)C3=CNC4=CC=CC=C43
10,000
5-HT1A
CORTEX
CN1C2CCC1CC(C2)OC(=O)C3=CNC4=CC=CC=C43
10,000
5-HT1A
CORTEX
null
2.33
5-HT1A
CORTEX
null
5.39
5-HT1A
CORTEX
C1CN=C(N1)C2COC3=CC=CC=C3O2
145.29
5-HT1A
CORTEX
C1CN=C(N1)C2COC3=CC=CC=C3O2
162.89
5-HT1A
CORTEX
CCN1C=CN=C1CC2COC3=CC=CC=C3O2
5,538.14
5-HT1A
CORTEX
CN(C)CCCN1C2=CC=CC=C2CCC3=CC=CC=C31
10,000
5-HT1A
HIPPOCAMPUS
CN(C)CCCN1C2=CC=CC=C2CCC3=CC=CC=C31
10,000
5-HT1A
HIPPOCAMPUS
COC1=CC2=C(C=C1)NC=C2C(CN)C(=O)OC.Cl
6.9
5-HT1A
HIPPOCAMPUS
COC1=CC2=C(C=C1)NC=C2C(CN)C(=O)OC.Cl
11.49
5-HT1A
CORTEX
C1CNCCC1CCC2=CNC3=CC=CC=C32
10,000
5-HT1A
HIPPOCAMPUS
C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O
1,933
5-HT1A
HIPPOCAMPUS
C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O
2,100
5-HT1A
CELLS
C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O
2,850
5-HT1A
BRAIN
C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O
3,243.33
5-HT1A
HIPPOCAMPUS
C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O
10,000
5-HT1A
CORTEX
CCN(CC)C(=O)NC1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
0.08
5-HT1A
CORTEX
CCN(CC)C(=O)NC1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
0.76
5-HT1A
CORTEX
CCN(CC)C(=O)NC1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
2.59
5-HT1A
HIPPOCAMPUS
CCN(CC)C(=O)NC1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
2.68
5-HT1A
HIPPO:LESIONED
CN1CCN(CC1)C2=NC3=CC=CC=C3OC4=C2C=C(C=C4)Cl
2,900
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
2.57
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
1.2
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
0.31
5-HT1A
HIPPOCAMPUS
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
0.64
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
2.05
5-HT1A
HIPPOCAMPUS
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
0.43
5-HT1A
HIPPOCAMPUS
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
2.57
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
3.9
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
4.1
5-HT1A
HIPPOCAMPUS
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
4.92
5-HT1A
CORTEX
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
5.47
5-HT1A
HIPPO:LESIONED
CCN(CC)C(=O)C1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C
10,000
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
3.45
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
3.7
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
4.34
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
5.52
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
7.63
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
7.94
5-HT1A
CORTEX
CN1CC(CC2C1CC3=CN(C4=CC=CC2=C34)C)CNC(=O)OCC5=CC=CC=C5
7.94
5-HT1A
CORTEX